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5YC8

Crystal structure of rationally thermostabilized M2 muscarinic acetylcholine receptor bound with NMS (Hg-derivative)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0005506molecular_functioniron ion binding
A0005886cellular_componentplasma membrane
A0007186biological_processG protein-coupled receptor signaling pathway
A0009055molecular_functionelectron transfer activity
A0016020cellular_componentmembrane
A0016907molecular_functionG protein-coupled acetylcholine receptor activity
A0020037molecular_functionheme binding
A0022900biological_processelectron transport chain
A0042597cellular_componentperiplasmic space
A0046872molecular_functionmetal ion binding
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues22
DetailsTRANSMEM: Helical; Name=1
ChainResidueDetails
AVAL23-MET45

site_idSWS_FT_FI2
Number of Residues55
DetailsTOPO_DOM: Cytoplasmic
ChainResidueDetails
AVAL46-ASN59
AASP120-MET139
ACYS443-ARG466

site_idSWS_FT_FI3
Number of Residues20
DetailsTRANSMEM: Helical; Name=2
ChainResidueDetails
ATYR60-TYR80

site_idSWS_FT_FI4
Number of Residues44
DetailsTOPO_DOM: Extracellular
ChainResidueDetails
ATHR81-ASP97
AGLN163-ALA184
ATHR411-PRO418

site_idSWS_FT_FI5
Number of Residues21
DetailsTRANSMEM: Helical; Name=3
ChainResidueDetails
ALEU98-PHE119

site_idSWS_FT_FI6
Number of Residues22
DetailsTRANSMEM: Helical; Name=4
ChainResidueDetails
AALA140-TRP162

site_idSWS_FT_FI7
Number of Residues24
DetailsTRANSMEM: Helical; Name=5
ChainResidueDetails
AALA185-ILE209

site_idSWS_FT_FI8
Number of Residues22
DetailsTRANSMEM: Helical; Name=6
ChainResidueDetails
ATHR388-ASN410

site_idSWS_FT_FI9
Number of Residues23
DetailsTRANSMEM: Helical; Name=7
ChainResidueDetails
AASN419-LEU442

site_idSWS_FT_FI10
Number of Residues3
DetailsMOD_RES: Phosphothreonine => ECO:0000255
ChainResidueDetails
ATHR446
ATHR450
ATHR465

site_idSWS_FT_FI11
Number of Residues2
DetailsBINDING: axial binding residue
ChainResidueDetails
ATRP1007
AILE1102

218853

PDB entries from 2024-04-24

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