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5YAW

Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction

Functional Information from GO Data
ChainGOidnamespacecontents
B0005095molecular_functionGTPase inhibitor activity
B0005515molecular_functionprotein binding
B0005737cellular_componentcytoplasm
B0005829cellular_componentcytosol
B0005929cellular_componentcilium
B0007601biological_processvisual perception
B0030659cellular_componentcytoplasmic vesicle membrane
B0031267molecular_functionsmall GTPase binding
B0031410cellular_componentcytoplasmic vesicle
B0050953biological_processsensory perception of light stimulus
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 8SL B 201
ChainResidue
BMET20
BLEU38
BSER39
BARG61
BLEU76
BGLN78
BILE109
BTHR131
BPHE133

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsRegion: {"description":"Required for association with membranes","evidences":[{"source":"PubMed","id":"9712853","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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