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5Y7Z

Complex structure of cyclin G-associated kinase with gefitinib

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue IRE A 401
ChainResidue
ALEU46
ALEU180
AALA67
ALYS69
AGLU124
ALEU125
ACYS126
ALYS127
AGLY128
AGLU132

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 402
ChainResidue
AARG157
AHIS161
AARG164

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 403
ChainResidue
AARG140
ASER207
AARG210
BARG140
BSER207
BARG210

site_idAC4
Number of Residues13
Detailsbinding site for residue IRE B 401
ChainResidue
BLEU46
BALA67
BLYS69
BGLU85
BGLU124
BLEU125
BCYS126
BLYS127
BGLY128
BGLU132
BLEU180
BCYS190
BASP191

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 B 402
ChainResidue
BHIS95
BARG157
BHIS161
BARG164

site_idAC6
Number of Residues3
Detailsbinding site for residue SO4 D 201
ChainResidue
DARG98
DARG99
DASN109

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 C 201
ChainResidue
AARG44
CARG98
CARG99
CASN109

Functional Information from PROSITE/UniProt
site_idPS00108
Number of Residues13
DetailsPROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. IiHrDLKveNLLL
ChainResidueDetails
AILE169-LEU181

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues548
DetailsDomain: {"description":"Protein kinase","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsActive site: {"description":"Proton acceptor","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"},{"source":"PROSITE-ProRule","id":"PRU10027","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

243531

PDB entries from 2025-10-22

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