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5XHE

Crystal structure analysis of the second bromodomain of BRD2 covalently linked to b-mercaptoethanol

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue PGE A 501
ChainResidue
ATRP370
AVAL435
AMET438
AGOL504
AHOH607

site_idAC2
Number of Residues8
Detailsbinding site for residue GOL A 502
ChainResidue
AASP444
AASP444
AGLU447
APHE448
ATYR426
AARG440
AGLN443
AGLN443

site_idAC3
Number of Residues6
Detailsbinding site for residue GOL A 503
ChainResidue
ALYS402
AASP407
AMET438
ALYS441
AHOH604
AHOH611

site_idAC4
Number of Residues5
Detailsbinding site for residue GOL A 504
ChainResidue
ALEU383
ACME425
AASN429
APGE501
AHOH603

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

223166

PDB entries from 2024-07-31

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