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5X0R

Crystal Structure of PXR LBD Complexed with SJB7

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue 4WH A 501
ChainResidue
AVAL211
ALEU428
APHE429
AMET243
ASER247
AALA280
APHE281
ATRP299
AHIS407
ATHR408
ALEU411

site_idAC2
Number of Residues10
Detailsbinding site for residue 4WH B 501
ChainResidue
BMET243
BALA280
BPHE281
BTRP299
BHIS407
BTHR408
BLEU411
BMET425
BLEU428
BPHE429

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
CSER698
DSER698
APRO384
BASN224
BSER262
BPRO384

222415

PDB entries from 2024-07-10

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