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5WR3

Thermolysin, SFX liganded form with water-based carrier

Functional Information from GO Data
ChainGOidnamespacecontents
A0004222molecular_functionmetalloendopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue NX6 A 401
ChainResidue
AASN112
ALEU202
AHIS231
AZN402
AHOH507
AHOH657
AALA113
ALEU133
AHIS142
AGLU143
AHIS146
ATYR157
AGLU166
AILE188

site_idAC2
Number of Residues5
Detailsbinding site for residue ZN A 402
ChainResidue
AHIS142
AHIS146
ATYR157
AGLU166
ANX6401

site_idAC3
Number of Residues6
Detailsbinding site for residue CA A 403
ChainResidue
AASP57
AASP59
AGLN61
AHOH533
AHOH546
AHOH692

site_idAC4
Number of Residues6
Detailsbinding site for residue CA A 404
ChainResidue
AASP138
AGLU177
AASP185
AGLU187
AGLU190
AHOH611

site_idAC5
Number of Residues6
Detailsbinding site for residue CA A 405
ChainResidue
AGLU177
AASN183
AASP185
AGLU190
AHOH553
AHOH576

site_idAC6
Number of Residues6
Detailsbinding site for residue CA A 406
ChainResidue
ATYR193
ATHR194
AILE197
AASP200
AHOH527
AHOH671

Functional Information from PROSITE/UniProt
site_idPS00142
Number of Residues10
DetailsZINC_PROTEASE Neutral zinc metallopeptidases, zinc-binding region signature. VVAHELTHAV
ChainResidueDetails
AVAL139-VAL148

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsActive site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU10095","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsActive site: {"description":"Proton donor","evidences":[{"source":"PROSITE-ProRule","id":"PRU10095","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues12
DetailsBinding site: {"evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues3
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU10095","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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