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5WIJ

JAK2 Pseudokinase in complex with NU6140

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue AQG A 901
ChainResidue
ALEU551
AGLY632
ALEU680
AHOH1047
AGLY552
AILE559
ALEU579
AGLN626
AGLU627
APHE628
AVAL629
ALYS630

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

222624

PDB entries from 2024-07-17

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