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5V7W

Crystal structure of human PARP14 bound to 2-{[(1-methylpiperidin-4-yl)methyl]amino}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 91J A 1901
ChainResidue
AHIS1682
AGLY1683
AASP1685
ATYR1714
AALA1716
ASER1722
ATHR1726
ATYR1727
AHOH2037

site_idAC2
Number of Residues9
Detailsbinding site for residue 91J B 1901
ChainResidue
BHIS1682
BGLY1683
BASP1685
BTYR1701
BTYR1714
BALA1716
BSER1722
BTYR1727
BHOH2011

246704

PDB entries from 2025-12-24

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