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5UT0

JAK2 JH2 in complex with AT9283

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue GOL A 901
ChainResidue
AASN673
ACYS675
AARG715
ATRP718

site_idAC2
Number of Residues4
Detailsbinding site for residue GOL A 902
ChainResidue
APHE694
AHOH1036
AHOH1101
AHOH1107

site_idAC3
Number of Residues13
Detailsbinding site for residue 35R A 903
ChainResidue
ALEU579
AGLU627
APHE628
AVAL629
ALYS630
APHE631
AGLY632
ALEU680
AHOH1009
AHOH1021
AHOH1077
AHOH1158
ALEU551

site_idAC4
Number of Residues3
Detailsbinding site for residue ACT A 904
ChainResidue
AGLY619
AASP620
AASN622

site_idAC5
Number of Residues1
Detailsbinding site for residue DMS A 905
ChainResidue
AASN782

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

225946

PDB entries from 2024-10-09

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