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5UC3

Structure of the dominant negative mutant Glucocorticoid Receptor alpha (L733K/N734P) complexed with RU-486

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 486 A 801
ChainResidue
AMET560
APHE623
AGLN642
AMET646
ACYS736
AHOH958
ALEU563
AASN564
AGLY567
AGLN570
ATRP600
AMET601
AMET604
AARG611

site_idAC2
Number of Residues5
Detailsbinding site for residue MPD A 802
ChainResidue
ATRP577
AMET604
AALA607
ALYS667
AHOH961

site_idAC3
Number of Residues4
Detailsbinding site for residue MPD A 803
ChainResidue
AHIS645
ATYR648
AGLU727
AASN731

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 804
ChainResidue
ASER617
AHIS654
AHOH909

site_idAC5
Number of Residues3
Detailsbinding site for residue EDO A 805
ChainResidue
ALYS743
ATHR744
AHOH976

site_idAC6
Number of Residues1
Detailsbinding site for residue EDO A 806
ChainResidue
AVAL658

site_idAC7
Number of Residues1
Detailsbinding site for residue EDO A 807
ChainResidue
AHOH938

site_idAC8
Number of Residues1
Detailsbinding site for residue EDO A 808
ChainResidue
APHE774

site_idAC9
Number of Residues3
Detailsbinding site for residue EDO A 809
ChainResidue
ATRP610
AARG614
AHOH984

site_idAD1
Number of Residues2
Detailsbinding site for residue EPE A 810
ChainResidue
APHE715
AHOH904

site_idAD2
Number of Residues10
Detailsbinding site for residue 486 B 801
ChainResidue
BMET560
BLEU563
BASN564
BGLY567
BGLN570
BTRP600
BARG611
BGLN642
BCYS736
BHOH910

site_idAD3
Number of Residues4
Detailsbinding site for residue MPD B 802
ChainResidue
BGLN570
BTRP577
BALA607
BLYS667

site_idAD4
Number of Residues2
Detailsbinding site for residue EDO B 803
ChainResidue
BHIS645
BASN731

site_idAD5
Number of Residues2
Detailsbinding site for residue EDO B 805
ChainResidue
BLYS743
BTHR744

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
ChainResidueDetails
ALYS703
BLYS703

237992

PDB entries from 2025-06-25

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