Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

5U6V

X-ray crystal structure of 1,2,3-triazolobenzodiazepine in complex with BRD2(D2)

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue 7WY A 501
ChainResidue
ATRP370
APRO371
APHE372
ALEU381
AASN429
AHIS433
AVAL435
AHOH604

site_idAC2
Number of Residues5
Detailsbinding site for residue EDO A 502
ChainResidue
AARG440
AASP444
AGLU447
AHOH601
ATYR426

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 503
ChainResidue
AILE389
AILE390
ALYS391
AHIS392
AASN424
ALYS427
AASP455

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 504
ChainResidue
ASER362
ALYS363
ALYS364

site_idAC5
Number of Residues3
Detailsbinding site for residue EDO A 505
ChainResidue
ALYS351
AASN354
AHOH602

site_idAC6
Number of Residues5
Detailsbinding site for residue EDO A 506
ChainResidue
ASER347
AGLU348
AGLN349
AHOH645
AHOH677

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

246031

PDB entries from 2025-12-10

PDB statisticsPDBj update infoContact PDBjnumon