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5U5M

CRYSTAL STRUCTURE OF I83E MEDITOPE-ENABLED TRASTUZUMAB WITH AZIDO-MEDITOPE

Functional Information from GO Data
ChainGOidnamespacecontents
C0019865molecular_functionimmunoglobulin binding
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue MRY B 301
ChainResidue
BGLU155
BPRO156
BVAL157
BALA175
BLEU185
BHOH435
BHOH456
D2GX5
DSER6

site_idAC2
Number of Residues32
Detailsbinding site for Ligand residues 56C D 8 through ARG D 9 bound to THR D 7
ChainResidue
AGLN38
ATHR40
AGLY42
ASER43
AGLU83
AALA84
AASP85
AHOH311
BVAL5
BGLU6
BSER7
BGLY9
BILE93
BTYR95
BGLN112
BGLY113
BTHR114
BLEU115
BPRO156
BLYS208
BPRO209
BHOH435
BHOH460
DPHE3
DASP4
D2GX5
DSER6
DTHR7
DLEU10
DARG11
DHOH101
DHOH103

site_idAC3
Number of Residues25
Detailsbinding site for Ligand 56C D 8 bound to THR D 7
ChainResidue
AGLN38
AGLY42
ASER43
BVAL5
BGLU6
BSER7
BGLY9
BILE93
BTYR95
BGLN112
BGLY113
BTHR114
BLEU115
BPRO156
BLYS208
BPRO209
BHOH435
BHOH460
DPHE3
DASP4
D2GX5
DSER6
DTHR7
DARG9
DHOH101

Functional Information from PROSITE/UniProt
site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. YACEVTH
ChainResidueDetails
ATYR192-HIS198
BTYR201-HIS207

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PDB entries from 2024-05-29

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