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5U2E

BRD4 first bromodomain (BD1) in complex with dual PI3 kinase (PI3K) inhibitor SF2535

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 837 A 201
ChainResidue
ATRP81
APRO82
AVAL87
ALYS91
AASN140
AHOH310
AHOH325

site_idAC2
Number of Residues9
Detailsbinding site for residue 837 B 201
ChainResidue
BVAL87
BLYS91
BLEU92
BASN140
BHOH315
BHOH320
BHOH360
BTRP81
BPRO82

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140
BASN140

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99
BLYS99

223532

PDB entries from 2024-08-07

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