5U2C
BRD4 second bromodomain (BD2) in complex with dual PI3 kinase (PI3K) inhibitor SF2558HA
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 7 |
Details | binding site for residue 82Y A 501 |
Chain | Residue |
A | TRP374 |
A | PRO375 |
A | VAL380 |
A | LEU385 |
A | TYR390 |
A | ASN433 |
A | HIS437 |
site_id | AC2 |
Number of Residues | 6 |
Details | binding site for residue 82Y B 501 |
Chain | Residue |
B | LEU385 |
B | TYR390 |
B | ASN433 |
B | HIS437 |
B | PRO375 |
B | VAL380 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | SITE: Acetylated histone binding => ECO:0000269|PubMed:22464331 |
Chain | Residue | Details |
A | ASN433 | |
B | ASN433 |