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5TWM

CRYSTAL STRUCTURE OF THE HEPATITIS C VIRUS GENOTYPE 2A STRAIN JFH1 L30S NS5B RNA-DEPENDENT RNA POLYMERASE IN COMPLEX WITH 5-[3-(tert-butylcarbamoyl)phenyl]-6-(ethylamino)-2-(4-fluorophenyl)-N-methylfuro[2,3-b]pyridine-3-carboxamide

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 7NG A 601
ChainResidue
AARG200
ALEU384
AGLN414
ATYR415
ATYR448
APHE551
AHOH767
ALEU204
ALEU314
AASP319
AVAL321
AILE363
ASER365
ACYS366
ASER368

site_idAC2
Number of Residues6
Detailsbinding site for residue SO4 A 602
ChainResidue
AASN24
AASN24
ASER27
ASER27
AHOH912
AHOH912

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 603
ChainResidue
AGLU446
AGLY449
AGLY556
AGLY557
AGLY558
AHOH777

site_idAC4
Number of Residues6
Detailsbinding site for residue SO4 A 604
ChainResidue
AGLU361
ASER371
AVAL372
ASER478
AHOH756
AHOH765

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 A 605
ChainResidue
AARG48
AARG158
AARG222
ACYS223

site_idAC6
Number of Residues9
Detailsbinding site for residue PE5 A 606
ChainResidue
ALYS100
ATYR101
APRO135
ATHR137
APHE267
AASN268
ASER269
AGLY271
AHOH808

site_idAC7
Number of Residues7
Detailsbinding site for residue PG4 A 607
ChainResidue
AGLU143
APHE145
ACYS146
ASER367
AARG386
ATHR390
AARG394

site_idAC8
Number of Residues9
Detailsbinding site for residue PG4 A 608
ChainResidue
ATRP6
AGLY8
AALA9
ASER46
AALA49
AALA209
AGLU210
ALYS211
AHOH927

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P26663
ChainResidueDetails
AASP220
AASP318
AASP319

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PDB entries from 2024-07-10

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