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5TEG

Crystal structure of hSETD8 in complex with histone H4K20 norleucine mutant peptide and S-Adenosylmethionine

Functional Information from GO Data
ChainGOidnamespacecontents
A0042799molecular_functionhistone H4K20 methyltransferase activity
B0042799molecular_functionhistone H4K20 methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue SAM A 401
ChainResidue
AGLY225
AHIS299
ATYR336
ATRP349
AHOH501
AHOH558
AHOH622
DHIS18
ALYS226
AARG228
ACYS270
ATYR271
AARG295
ALEU296
AILE297
AASN298

site_idAC2
Number of Residues20
Detailsbinding site for residue SAM B 401
ChainResidue
AHOH615
BGLY225
BLYS226
BARG228
BCYS270
BTYR271
BARG295
BLEU296
BILE297
BASN298
BHIS299
BTYR336
BTRP349
BHOH509
BHOH546
BHOH551
BHOH573
BHOH587
BHOH619
EHIS18

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsDNA_BIND:
ChainResidueDetails
DLYS16-NLE20
ELYS16-NLE20
AASN298
BLYS226
BTYR271
BASN298

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: N6-propionyllysine; alternate => ECO:0000269|PubMed:17267393
ChainResidueDetails
DLYS16
ELYS16

site_idSWS_FT_FI3
Number of Residues2
DetailsMOD_RES: N6-methyllysine; alternate => ECO:0000269|PubMed:12086618, ECO:0000269|PubMed:15964846, ECO:0000269|PubMed:17967882, ECO:0000269|PubMed:27338793
ChainResidueDetails
DNLE20
ENLE20

site_idSWS_FT_FI4
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2); alternate => ECO:0007744|PubMed:28112733
ChainResidueDetails
DNLE20
ENLE20

222624

PDB entries from 2024-07-17

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