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5TCM

First Bromodomain from Leishmania donovani LdBPK.091320 complexed with BI-2536

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue R78 A 201
ChainResidue
AHIS23
AHOH341
CTHR33
CTYR34
CR78200
AHIS24
AILE25
AVAL30
ATYR86
AASN87
ATYR93
AHOH302
AHOH309

site_idAC2
Number of Residues9
Detailsbinding site for residue EDO A 202
ChainResidue
ALEU17
AASP18
AARG19
AASP22
AHIS24
AILE25
APHE26
AALA27
APHE100

site_idAC3
Number of Residues10
Detailsbinding site for residue R78 B 201
ChainResidue
BHIS23
BHIS24
BILE25
BVAL30
BTYR34
BTYR86
BASN87
BTYR93
BHOH304
BHOH305

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO B 202
ChainResidue
BTYR36
BALA38
BGLU39

site_idAC5
Number of Residues5
Detailsbinding site for residue EDO B 203
ChainResidue
BLYS99
BARG102
BTYR103
BGLU106
BHOH370

site_idAC6
Number of Residues12
Detailsbinding site for residue R78 C 200
ChainResidue
ATYR34
AR78201
CHIS24
CILE25
CVAL30
CTHR33
CTYR86
CASN87
CTYR93
CHOH304
CHOH309
CHOH315

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PDB entries from 2024-06-12

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