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5T4U

Crystal structure of the bromodomain of human BRPF1 in complex with a quinolinone ligand

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue NO3 A 801
ChainResidue
ASER702
ALEU705
ALYS706
ATYR715
AVAL719
AARG722
AHOH948

site_idAC2
Number of Residues6
Detailsbinding site for residue 12Q A 802
ChainResidue
APRO658
AASN708
APHE714
AHOH906
AILE652
AVAL657

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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