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5Q0Q

Ligand binding to FARNESOID-X-RECEPTOR

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
A0032052molecular_functionbile acid binding
A0038183biological_processbile acid signaling pathway
C0003677molecular_functionDNA binding
C0004879molecular_functionnuclear receptor activity
C0006355biological_processregulation of DNA-templated transcription
C0032052molecular_functionbile acid binding
C0038183biological_processbile acid signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 9LD A 501
ChainResidue
AMET269
ASER336
AILE339
ALEU352
AILE356
ATYR373
AHIS451
AMET454
ATRP473
ALEU291
ATHR292
AMET294
AALA295
AASN297
AHIS298
AMET332
AARG335

site_idAC2
Number of Residues15
Detailsbinding site for residue 9LD C 501
ChainResidue
CMET269
CPHE288
CTHR292
CMET294
CALA295
CASN297
CHIS298
CVAL301
CSER336
CILE339
CLEU352
CTYR373
CHIS451
CPHE465
CTRP473

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBinding site: {"evidences":[{"source":"PDB","id":"6HL1","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphothreonine; by PKC/PRKCZ","evidences":[{"source":"PubMed","id":"18668687","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO1)","evidences":[{"source":"PubMed","id":"23546875","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 5"}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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