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5OWE

Crystal structure of the human BRPF1 bromodomain in complex with DSPBP1010

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue B0E A 801
ChainResidue
AILE652
AVAL657
AVAL662
AASN708
APHE714
AHOH913
AHOH916
AHOH920

site_idAC2
Number of Residues7
Detailsbinding site for residue NO3 A 802
ChainResidue
ALEU705
ALYS706
ATYR715
AARG722
AHOH936
AHOH946
ASER702

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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