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5OWB

Crystal structure of the human BRPF1 bromodomain in complex with DSPBP1004

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue NO3 A 801
ChainResidue
ASER702
ALEU705
ALYS706
ATYR715
AARG722
AHOH967

site_idAC2
Number of Residues11
Detailsbinding site for residue AYW A 802
ChainResidue
AVAL662
ATYR707
AASN708
APHE714
AHOH912
AHOH917
AHOH973
AHOH994
AILE652
AVAL657
APRO658

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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