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5OVE

Ras guanine nucleotide exchange factor SOS1 (Rem-cdc25) in complex with small molecule inhibitor compound 1

Functional Information from GO Data
ChainGOidnamespacecontents
A0005085molecular_functionguanyl-nucleotide exchange factor activity
A0007264biological_processsmall GTPase-mediated signal transduction
Functional Information from PDB Data
site_idAC1
Number of Residues2
Detailsbinding site for residue EDO A 1101
ChainResidue
AGLU565
AGLU680

site_idAC2
Number of Residues5
Detailsbinding site for residue EDO A 1102
ChainResidue
AARG786
AGLU864
APRO1042
AHOH1338
AHOH1358

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 1103
ChainResidue
ATYR1031
AHOH1299
AASP775
ACYS838

site_idAC4
Number of Residues10
Detailsbinding site for residue AXE A 1104
ChainResidue
AMET878
AASN879
ATYR884
APHE890
ALYS898
ALEU901
AGLU902
AHIS905
AARG950
AHOH1302

Functional Information from PROSITE/UniProt
site_idPS00720
Number of Residues34
DetailsRASGEF Ras Guanine-nucleotide exchange factors domain signature. VPFfGiyLtNIlkteegnpevlkrhgkel.................INFsK
ChainResidueDetails
AVAL927-LYS960

219140

PDB entries from 2024-05-01

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