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5OVB

Crystal structure of human BRD4(1) bromodomain in complex with DR46

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue AY2 A 201
ChainResidue
ATRP81
AHOH396
APRO82
AGLN85
AVAL87
AASN140
AILE146
AHOH312
AHOH330
AHOH388

site_idAC2
Number of Residues11
Detailsbinding site for residue AY2 B 201
ChainResidue
ATRP81
BTRP81
BPRO82
BGLN85
BLEU92
BASN140
BILE146
BHOH331
BHOH358
BHOH372
BHOH382

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140
BASN140

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99
BLYS99

222624

PDB entries from 2024-07-17

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