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5OIA

Dissociation of biochemical and antiretroviral activities of Integrase-LEDGF Allosteric Inhibitors revealed by resistance of A125 polymorphic HIV-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue MG A 301
ChainResidue
AASP64
ACAS65
AASN120

site_idAC2
Number of Residues4
Detailsbinding site for residue MG A 302
ChainResidue
ASER123
AALA125
AHOH435
AHOH441

site_idAC3
Number of Residues10
Detailsbinding site for residue 9VK A 303
ChainResidue
AALA128
ATRP132
AALA169
AGLU170
AHIS171
ATHR174
AHOH414
AHOH428
AGLN95
AALA125

site_idAC4
Number of Residues4
Detailsbinding site for residue SO4 A 304
ChainResidue
ALYS71
AHIS171
ALEU172
AHOH408

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P04585","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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