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5O5H

Crystal structure of the human BRPF1 bromodomain in complex with BZ053

Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue 9LK A 801
ChainResidue
APHE653
A9LK802
AHOH925
AVAL657
APRO658
AVAL662
ACYS704
ATYR707
AASN708
APHE714
ALYS738

site_idAC2
Number of Residues11
Detailsbinding site for residue 9LK A 802
ChainResidue
APHE653
AVAL657
AGLU661
AVAL662
ATYR707
AASN708
APHE714
ALYS738
A9LK801
AHOH910
AHOH925

site_idAC3
Number of Residues9
Detailsbinding site for residue NO3 A 803
ChainResidue
ASER702
ALEU705
ALEU705
ALYS706
ATYR715
AVAL719
AARG722
AHOH955
AHOH966

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

218853

PDB entries from 2024-04-24

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