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5NOB

Crystal structure of human tankyrase 2 in complex with OD336

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 92T A 1301
ChainResidue
AHIS1031
ATYR1071
AILE1075
AHOH1433
AHOH1438
ASER1033
APHE1035
AILE1039
APHE1044
AASP1045
AHIS1048
ATYR1050
ATYR1060

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 1302
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC3
Number of Residues13
Detailsbinding site for residue 92T B 1301
ChainResidue
BHIS1031
BSER1033
BPHE1035
BILE1039
BPHE1044
BASP1045
BHIS1048
BTYR1050
BTYR1060
BTYR1071
BHOH1423
BHOH1438
BHOH1459

site_idAC4
Number of Residues4
Detailsbinding site for residue ZN B 1302
ChainResidue
BCYS1081
BHIS1084
BCYS1089
BCYS1092

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
BCYS1081
BHIS1084
BCYS1089
BCYS1092

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PDB entries from 2024-07-10

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