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5NIQ

exendin-4 variant with dual GLP-1 / glucagon receptor activity

Functional Information from GO Data
ChainGOidnamespacecontents
A0005179molecular_functionhormone activity
A0005576cellular_componentextracellular region
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue D6M A 101
ChainResidue
ALYS14
AARG17
AARG18

site_idAC2
Number of Residues1
Detailsbinding site for Ligand NH2 A 40 bound to SER A 39
ChainResidue
ASER39

Functional Information from PROSITE/UniProt
site_idPS00260
Number of Residues23
DetailsGLUCAGON Glucagon / GIP / secretin / VIP family signature. HSQGTFtSDLskqkdsrrAQDFI
ChainResidueDetails
AHIS1-ILE23

248335

PDB entries from 2026-01-28

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