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5N8V

Targeting the PEX14-PEX5 interaction by small molecules provides novel therapeutic routes to treat trypanosomiases.

Functional Information from GO Data
ChainGOidnamespacecontents
A0005778cellular_componentperoxisomal membrane
A0016560biological_processprotein import into peroxisome matrix, docking
B0005778cellular_componentperoxisomal membrane
B0016560biological_processprotein import into peroxisome matrix, docking
D0005778cellular_componentperoxisomal membrane
D0016560biological_processprotein import into peroxisome matrix, docking
F0005778cellular_componentperoxisomal membrane
F0016560biological_processprotein import into peroxisome matrix, docking
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue KZZ A 101
ChainResidue
AASN13
AHOH232
AHOH243
FHIS33
FPHE34
FKZZ101
AGLU16
APHE17
ATHR26
APHE34
ALEU35
ALYS38
AHOH225
AHOH229

site_idAC2
Number of Residues7
Detailsbinding site for residue SO4 A 102
ChainResidue
ASER5
AGLU6
AHOH204
AHOH223
AHOH241
BSER41
BALA42

site_idAC3
Number of Residues7
Detailsbinding site for residue SO4 A 103
ChainResidue
ASER41
AALA42
AHOH230
AHOH235
AHOH244
BSER5
BGLU6

site_idAC4
Number of Residues5
Detailsbinding site for residue SO4 A 104
ChainResidue
APRO27
ATHR28
AHOH201
AHOH206
AHOH214

site_idAC5
Number of Residues3
Detailsbinding site for residue BME A 105
ChainResidue
AGLU43
ACYS46
AHOH257

site_idAC6
Number of Residues2
Detailsbinding site for residue CL A 106
ChainResidue
AHIS33
FARG25

site_idAC7
Number of Residues14
Detailsbinding site for residue KZZ B 101
ChainResidue
BASN13
BGLU16
BPHE17
BTHR26
BPHE34
BLEU35
BLYS38
BHOH210
BHOH227
BHOH230
DHIS33
DPHE34
DKZZ101
DHOH267

site_idAC8
Number of Residues6
Detailsbinding site for residue SO4 B 102
ChainResidue
BTHR57
BASN59
BARG63
BHOH236
DBME104
DHOH244

site_idAC9
Number of Residues3
Detailsbinding site for residue BME B 103
ChainResidue
BGLU43
BCYS46
BTHR50

site_idAD1
Number of Residues1
Detailsbinding site for residue CL B 104
ChainResidue
BTHR28

site_idAD2
Number of Residues14
Detailsbinding site for residue KZZ D 101
ChainResidue
BSER30
BHIS33
BPHE34
BSER37
BKZZ101
DASN13
DGLU16
DPHE17
DTHR26
DPHE34
DLEU35
DLYS38
DHOH216
DHOH232

site_idAD3
Number of Residues6
Detailsbinding site for residue SO4 D 102
ChainResidue
DPRO27
DTHR28
DSER29
DHOH203
DHOH208
DHOH224

site_idAD4
Number of Residues6
Detailsbinding site for residue SO4 D 103
ChainResidue
DTHR57
DASN59
DARG63
DHOH205
DHOH212
DHOH225

site_idAD5
Number of Residues5
Detailsbinding site for residue BME D 104
ChainResidue
BTHR57
BSO4102
DCYS46
DGLU47
DTHR50

site_idAD6
Number of Residues16
Detailsbinding site for residue KZZ F 101
ChainResidue
FGLU16
FPHE17
FARG22
FTHR26
FPHE34
FLEU35
FLYS38
FHOH226
FHOH227
FHOH237
AHIS33
APHE34
ASER37
AKZZ101
FASN13
FALA14

site_idAD7
Number of Residues3
Detailsbinding site for residue BME F 102
ChainResidue
AASN59
FCYS46
FHOH209

223166

PDB entries from 2024-07-31

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