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5N49

BRPF2 in complex with Compound 7

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 8LW B 701
ChainResidue
ALEU562
BASN642
BPHE648
BHOH810
BHOH816
AASP645
ATHR646
BALA584
BILE586
BGLN589
BVAL591
BSER592
BTYR641

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AriFaqpvSlkevp..DYLdhIkhpMdfatMrkrleaqg..Yknlhefeedfdl.IidNCmkY
ChainResidueDetails
AALA584-TYR641

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues208
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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