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5N2L

Crystal structure of the second bromodomain of human BRD2 in complex with a tetrahydroquinoline analogue

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue SO4 A 501
ChainResidue
AHIS365
AVAL445
AARG449
CARG440

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 502
ChainResidue
ASER362
ALYS363
ALYS364
AHOH648

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 503
ChainResidue
CMET394
CLYS402
ASER379

site_idAC4
Number of Residues16
Detailsbinding site for residue 8J2 A 504
ChainResidue
ATRP370
APRO371
APHE372
ALEU383
ACYS425
AASN429
AHIS433
AVAL435
AHOH604
AHOH607
AHOH615
AHOH637
AHOH659
BLYS363
BTRP370
BTYR373

site_idAC5
Number of Residues5
Detailsbinding site for residue SO4 B 501
ChainResidue
BLYS364
BHIS365
BARG440
BARG449
BHOH628

site_idAC6
Number of Residues5
Detailsbinding site for residue SO4 B 502
ChainResidue
BVAL376
BASP377
BALA378
BSER379
BHIS387

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 B 503
ChainResidue
BSER362
BLYS363
BHIS384
BHOH620

site_idAC8
Number of Residues15
Detailsbinding site for residue 8J2 B 504
ChainResidue
ALYS363
ATYR373
AHOH630
BTRP370
BPRO371
BPHE372
BLEU381
BLEU383
BCYS425
BASN429
BHIS433
BMET438
BHOH615
BHOH639
BHOH640

site_idAC9
Number of Residues4
Detailsbinding site for residue SO4 C 501
ChainResidue
AARG440
CLYS364
CHIS365
CARG449

site_idAD1
Number of Residues4
Detailsbinding site for residue EDO C 502
ChainResidue
CVAL376
CALA378
CSER379
CHIS387

site_idAD2
Number of Residues14
Detailsbinding site for residue 8J2 C 503
ChainResidue
CTRP370
CPRO371
CPHE372
CLEU383
CCYS425
CASN429
CHIS433
CASP434
CMET438
CHOH605
CHOH634
CHOH665
DLYS363
DTYR373

site_idAD3
Number of Residues13
Detailsbinding site for residue 8J2 C 504
ChainResidue
CTYR373
CHOH639
CHOH647
CHOH648
DTRP370
DPRO371
DPHE372
DLEU383
DCYS425
DASN429
DHIS433
DMET438
DHOH617

site_idAD4
Number of Residues5
Detailsbinding site for residue SO4 D 501
ChainResidue
DLYS364
DHIS365
DARG440
DVAL445
DARG449

site_idAD5
Number of Residues3
Detailsbinding site for residue EDO D 502
ChainResidue
DALA437
DLYS441
DHOH601

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

218853

PDB entries from 2024-04-24

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