Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 4 |
| Details | binding site for residue SO4 A 501 |
| Chain | Residue |
| A | HIS365 |
| A | VAL445 |
| A | ARG449 |
| C | ARG440 |
| site_id | AC2 |
| Number of Residues | 4 |
| Details | binding site for residue EDO A 502 |
| Chain | Residue |
| A | SER362 |
| A | LYS363 |
| A | LYS364 |
| A | HOH648 |
| site_id | AC3 |
| Number of Residues | 3 |
| Details | binding site for residue EDO A 503 |
| Chain | Residue |
| C | MET394 |
| C | LYS402 |
| A | SER379 |
| site_id | AC4 |
| Number of Residues | 16 |
| Details | binding site for residue 8J2 A 504 |
| Chain | Residue |
| A | TRP370 |
| A | PRO371 |
| A | PHE372 |
| A | LEU383 |
| A | CYS425 |
| A | ASN429 |
| A | HIS433 |
| A | VAL435 |
| A | HOH604 |
| A | HOH607 |
| A | HOH615 |
| A | HOH637 |
| A | HOH659 |
| B | LYS363 |
| B | TRP370 |
| B | TYR373 |
| site_id | AC5 |
| Number of Residues | 5 |
| Details | binding site for residue SO4 B 501 |
| Chain | Residue |
| B | LYS364 |
| B | HIS365 |
| B | ARG440 |
| B | ARG449 |
| B | HOH628 |
| site_id | AC6 |
| Number of Residues | 5 |
| Details | binding site for residue SO4 B 502 |
| Chain | Residue |
| B | VAL376 |
| B | ASP377 |
| B | ALA378 |
| B | SER379 |
| B | HIS387 |
| site_id | AC7 |
| Number of Residues | 4 |
| Details | binding site for residue SO4 B 503 |
| Chain | Residue |
| B | SER362 |
| B | LYS363 |
| B | HIS384 |
| B | HOH620 |
| site_id | AC8 |
| Number of Residues | 15 |
| Details | binding site for residue 8J2 B 504 |
| Chain | Residue |
| A | LYS363 |
| A | TYR373 |
| A | HOH630 |
| B | TRP370 |
| B | PRO371 |
| B | PHE372 |
| B | LEU381 |
| B | LEU383 |
| B | CYS425 |
| B | ASN429 |
| B | HIS433 |
| B | MET438 |
| B | HOH615 |
| B | HOH639 |
| B | HOH640 |
| site_id | AC9 |
| Number of Residues | 4 |
| Details | binding site for residue SO4 C 501 |
| Chain | Residue |
| A | ARG440 |
| C | LYS364 |
| C | HIS365 |
| C | ARG449 |
| site_id | AD1 |
| Number of Residues | 4 |
| Details | binding site for residue EDO C 502 |
| Chain | Residue |
| C | VAL376 |
| C | ALA378 |
| C | SER379 |
| C | HIS387 |
| site_id | AD2 |
| Number of Residues | 14 |
| Details | binding site for residue 8J2 C 503 |
| Chain | Residue |
| C | TRP370 |
| C | PRO371 |
| C | PHE372 |
| C | LEU383 |
| C | CYS425 |
| C | ASN429 |
| C | HIS433 |
| C | ASP434 |
| C | MET438 |
| C | HOH605 |
| C | HOH634 |
| C | HOH665 |
| D | LYS363 |
| D | TYR373 |
| site_id | AD3 |
| Number of Residues | 13 |
| Details | binding site for residue 8J2 C 504 |
| Chain | Residue |
| C | TYR373 |
| C | HOH639 |
| C | HOH647 |
| C | HOH648 |
| D | TRP370 |
| D | PRO371 |
| D | PHE372 |
| D | LEU383 |
| D | CYS425 |
| D | ASN429 |
| D | HIS433 |
| D | MET438 |
| D | HOH617 |
| site_id | AD4 |
| Number of Residues | 5 |
| Details | binding site for residue SO4 D 501 |
| Chain | Residue |
| D | LYS364 |
| D | HIS365 |
| D | ARG440 |
| D | VAL445 |
| D | ARG449 |
| site_id | AD5 |
| Number of Residues | 3 |
| Details | binding site for residue EDO D 502 |
| Chain | Residue |
| D | ALA437 |
| D | LYS441 |
| D | HOH601 |
Functional Information from PROSITE/UniProt
| site_id | PS00633 |
| Number of Residues | 60 |
| Details | BROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY |
| Chain | Residue | Details |
| A | ALA369-TYR428 | |