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5N17

First Bromodomain (BD1) from Candida albicans Bdf1 bound to a dibenzothiazepinone (compound 3)

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue 8FK A 401
ChainResidue
APRO233
APHE234
APHE290
AASN291
AILE297
AHOH505

site_idAC2
Number of Residues6
Detailsbinding site for residue SO4 A 402
ChainResidue
AHOH510
BLYS288
BGLU293
AALA190
ALYS289
AHOH506

site_idAC3
Number of Residues3
Detailsbinding site for residue SO4 A 403
ChainResidue
AGLY296
AHOH512
AHOH536

site_idAC4
Number of Residues6
Detailsbinding site for residue 8FK B 401
ChainResidue
BPRO233
BPHE234
BPHE290
BASN291
BHOH514
BHOH603

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AvpFlhpvDtvklnvpFYYnyIprpMdlstIerkinlka..Yedvsqvvddfnl.MvkNCkkF
ChainResidueDetails
AALA231-PHE290

222415

PDB entries from 2024-07-10

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