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5MWH

Crystal structure of the human BRPF1 bromodomain in complex with BZ089

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue UWX A 801
ChainResidue
AILE652
AHOH903
AHOH911
AHOH918
AHOH943
BLYS639
APHE653
AVAL657
APRO658
AGLU661
ACYS704
ATYR707
AASN708
APHE714

site_idAC2
Number of Residues13
Detailsbinding site for residue UWX B 801
ChainResidue
ALYS639
BILE652
BPHE653
BVAL657
BPRO658
BGLU661
BCYS704
BTYR707
BASN708
BPHE714
BHOH903
BHOH919
BHOH922

site_idAC3
Number of Residues6
Detailsbinding site for residue NO3 B 802
ChainResidue
BLEU630
BTHR631
BLEU634
BILE635
BARG638
BHOH954

site_idAC4
Number of Residues7
Detailsbinding site for residue NO3 B 803
ChainResidue
AASP691
AGLU694
AARG733
AHOH931
BGLU694
BLEU729
BARG733

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

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PDB entries from 2024-07-24

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