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5MQK

Crystal structure of CREBBP bromodomain complexed with CBP019

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue QPR A 1201
ChainResidue
APRO1110
AVAL1115
AASN1168
AVAL1174
AHOH1318

site_idAC2
Number of Residues4
Detailsbinding site for residue QPR B 1201
ChainResidue
BPRO1110
BVAL1115
BASN1168
BHOH1325

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-07-24

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