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5MPK

Crystal structure of CREBBP bromodomain complexed with DK19

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 0BC A 1201
ChainResidue
ALEU1109
APRO1110
AGLN1113
AVAL1115
ALEU1120
AASN1168
AARG1173
AHOH1306
AHOH1313

site_idAC2
Number of Residues10
Detailsbinding site for residue 0BC B 1201
ChainResidue
ATRP1165
BPRO1110
BVAL1115
BLEU1120
BASN1168
BARG1173
BVAL1174
BHOH1306
BHOH1309
BHOH1331

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-04-17

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