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5MKX

1.68A STRUCTURE PCAF BROMODOMAIN WITH 4-chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
B0004402molecular_functionhistone acetyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 82I A 901
ChainResidue
APRO747
AVAL752
AGLU756
ATYR802
AASN803
ATYR809
AHOH1020

site_idAC2
Number of Residues8
Detailsbinding site for residue SO4 A 902
ChainResidue
AHOH1014
AHOH1029
AHOH1066
BTYR729
BARG780
BHOH1019
AARG776
AHOH1001

site_idAC3
Number of Residues8
Detailsbinding site for residue EPE A 903
ChainResidue
APRO751
AARG754
ATYR761
AHOH1062
AHOH1063
AHOH1074
AHOH1144
BHOH1004

site_idAC4
Number of Residues6
Detailsbinding site for residue 82I B 901
ChainResidue
BPRO747
BPHE748
BTYR802
BASN803
BTYR809
BHOH1008

site_idAC5
Number of Residues1
Detailsbinding site for residue BU1 B 902
ChainResidue
BPHE766

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFmepvKrteap..GYYevIrfpMdlktMserlknry..Yvskklfmadlqr.VftNCkeY
ChainResidueDetails
AALA745-TYR802

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PDB entries from 2024-07-10

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