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5M6M

Small Molecule inhibitors of IAP

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues7
Detailsbinding site for residue NA A 402
ChainResidue
AHOH553
AHOH553
ATHR271
APHE272
APHE272
ATHR274
AHOH504

site_idAC3
Number of Residues11
Detailsbinding site for residue 7H8 A 403
ChainResidue
AVAL298
AGLY306
ALEU307
ATHR308
AASP309
ATRP310
AGLU314
AGLN319
ATRP323
ATYR324
AHOH513

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues66
DetailsBIR_REPEAT_1 BIR repeat. YeaRiftfgt.Wiysvnkeqlar...AGFyAlgegDkvkCfhCgggltdWkpsedpweqHakwyPgCkyL
ChainResidueDetails
ATYR265-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00029
ChainResidueDetails
ACYS300
ACYS303
AHIS320
ACYS327

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:12747801
ChainResidueDetails
ALYS322
ALYS328

219140

PDB entries from 2024-05-01

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