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5KTU

Crystal structure of the bromodomain of human CREBBP bound to pyrazolopiperidine scaffold

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 6XB A 1201
ChainResidue
APRO1110
AVAL1115
AASN1168
AHOH1307
AHOH1324
AHOH1326
BARG1112

site_idAC2
Number of Residues4
Detailsbinding site for residue DMS B 1201
ChainResidue
BASN1168
BHOH1308
BPRO1110
BVAL1115

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

222624

PDB entries from 2024-07-17

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