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5KRS

HIV-1 Integrase Catalytic Core Domain in Complex with an Allosteric Inhibitor, 3-(1H-pyrrol-1-yl)-2-thiophenecarboxylic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues1
Detailsbinding site for residue DMS A 301
ChainResidue
ATRP131

site_idAC2
Number of Residues12
Detailsbinding site for residue 6XI A 302
ChainResidue
AHOH419
AHOH448
AHOH467
AHOH485
ACAF65
AGLU92
ATHR93
AGLY94
ASER119
AASN120
ATHR122
ASER123

site_idAC3
Number of Residues3
Detailsbinding site for residue 6XI A 303
ChainResidue
AGLU170
AHOH401
AHOH438

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P04585","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

242500

PDB entries from 2025-10-01

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