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5KRE

Covalent inhibitor of LYPLAL1

Functional Information from GO Data
ChainGOidnamespacecontents
A0004622molecular_functionphosphatidylcholine lysophospholipase activity
A0005515molecular_functionprotein binding
A0005737cellular_componentcytoplasm
A0005739cellular_componentmitochondrion
A0005829cellular_componentcytosol
A0008474molecular_functionpalmitoyl-(protein) hydrolase activity
A0016298molecular_functionlipase activity
A0016787molecular_functionhydrolase activity
A0016788molecular_functionhydrolase activity, acting on ester bonds
A0042997biological_processnegative regulation of Golgi to plasma membrane protein transport
A0098734biological_processmacromolecule depalmitoylation
A0160049biological_processnegative regulation of cGAS/STING signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 6WG A 301
ChainResidue
ASER30
AHOH427
ATYR66
AARG80
AILE83
ASER124
AMET125
ALEU181
AVAL182
ANO3302

site_idAC2
Number of Residues9
Detailsbinding site for residue NO3 A 302
ChainResidue
AARG80
ASER124
AMET125
ACYS128
ASER148
ASER149
APHE150
AVAL182
A6WG301

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsActive site: {"description":"Charge relay system","evidences":[{"source":"UniProtKB","id":"O75608","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsActive site: {"description":"Charge relay system","evidences":[{"source":"PubMed","id":"37802025","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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