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5KM5

Human Histidine Triad Nucleotide Binding Protein 2 (hHint2) triciribine 5'-monoposphate catalytic product complex

Functional Information from GO Data
ChainGOidnamespacecontents
A0003824molecular_functioncatalytic activity
B0003824molecular_functioncatalytic activity
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue CL A 201
ChainResidue
AASN136
ASER144
AHIS151

site_idAC2
Number of Residues6
Detailsbinding site for residue PG4 A 202
ChainResidue
AARG156
AGLN159
BGLN73
BGLN74
BLYS95
BGLY163

site_idAC3
Number of Residues19
Detailsbinding site for residue TR5 B 201
ChainResidue
APRO93
ALYS94
AHIS147
BPHE56
BILE59
BLEU64
BPHE78
BARG79
BASP80
BVAL81
BALA82
BASN136
BALA142
BSER144
BVAL145
BHIS149
BHIS151
BHOH310
BHOH312

Functional Information from PROSITE/UniProt
site_idPS00892
Number of Residues19
DetailsHIT_1 HIT domain signature. NdgklGaQsVyHLHIHVLG
ChainResidueDetails
AASN136-GLY154

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Tele-AMP-histidine intermediate => ECO:0000269|PubMed:16762638
ChainResidueDetails
AHIS149
BHIS149

site_idSWS_FT_FI2
Number of Residues10
DetailsBINDING: BINDING => ECO:0000269|PubMed:23659632, ECO:0007744|PDB:4INI
ChainResidueDetails
ASER63
BHIS149
AASP80
AASN136
AALA142
AHIS149
BSER63
BASP80
BASN136
BALA142

site_idSWS_FT_FI3
Number of Residues4
DetailsMOD_RES: N6-acetyllysine => ECO:0000250|UniProtKB:Q9D0S9
ChainResidueDetails
ALYS119
ALYS139
BLYS119
BLYS139

218853

PDB entries from 2024-04-24

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