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5KE2

Crystal structure of SETDB1 Tudor domain in complex with inhibitor XST06472A

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue 6S4 A 501
ChainResidue
ATRP358
ATRP363
APHE379
AASP382
AARG384
ACYS385

site_idAC2
Number of Residues8
Detailsbinding site for residue EDO A 502
ChainResidue
ATHR320
AHOH611
AHOH634
AHOH662
AHOH737
ATYR193
ASER262
APRO316

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 503
ChainResidue
AGLU322
AARG330
ALEU348
ALYS349
AHOH616
AHOH618

site_idAC4
Number of Residues6
Detailsbinding site for residue SO4 A 504
ChainResidue
AARG209
ATRP363
ALYS364
AASP381
AHOH612
AHOH719

site_idAC5
Number of Residues7
Detailsbinding site for residue SO4 A 505
ChainResidue
AHIS214
ALYS215
AHOH609
AHOH615
AHOH621
AHOH646
AHOH686

site_idAC6
Number of Residues8
Detailsbinding site for residue SO4 A 506
ChainResidue
ALYS229
ALEU242
ASER243
AHIS246
AHOH602
AHOH625
AHOH679
AHOH690

site_idAC7
Number of Residues4
Detailsbinding site for residue SO4 A 507
ChainResidue
ATHR306
AGLN307
ASER308
AARG384

site_idAC8
Number of Residues6
Detailsbinding site for residue SO4 A 508
ChainResidue
AGLU357
AGLY360
ATRP362
APHE399
AHOH721
AHOH767

site_idAC9
Number of Residues2
Detailsbinding site for residue SO4 A 509
ChainResidue
AARG203
ALYS215

223166

PDB entries from 2024-07-31

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