5JTY
Glutamate- and DCKA-bound GluN1/GluN2A agonist binding domains with MPX-007
Functional Information from GO Data
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 10 |
Details | binding site for residue 2JK A 501 |
Chain | Residue |
A | GLN13 |
A | PHE250 |
A | PHE16 |
A | PHE92 |
A | PRO124 |
A | LEU125 |
A | THR126 |
A | ARG131 |
A | TRP223 |
A | VAL227 |
site_id | AC2 |
Number of Residues | 14 |
Details | binding site for residue 6ND B 601 |
Chain | Residue |
A | PRO140 |
A | ARG247 |
A | SER248 |
A | GLY249 |
B | VAL129 |
B | PRO130 |
B | PHE131 |
B | VAL132 |
B | GLU133 |
B | LEU264 |
B | VAL267 |
B | MET272 |
B | GLU276 |
B | LEU280 |
site_id | AC3 |
Number of Residues | 11 |
Details | binding site for residue GLU B 602 |
Chain | Residue |
B | HIS88 |
B | SER114 |
B | LEU115 |
B | THR116 |
B | ARG121 |
B | GLY172 |
B | SER173 |
B | THR174 |
B | TYR214 |
B | ASP215 |
B | HOH705 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | BINDING: BINDING => ECO:0000269|PubMed:16281028, ECO:0007744|PDB:2A5S, ECO:0007744|PDB:2A5T, ECO:0007744|PDB:4NF4, ECO:0007744|PDB:4NF8, ECO:0007744|PDB:5I56, ECO:0007744|PDB:5I57, ECO:0007744|PDB:5I58, ECO:0007744|PDB:5I59, ECO:0007744|PDB:5JTY |
Chain | Residue | Details |
B | SER114 |
site_id | SWS_FT_FI2 |
Number of Residues | 1 |
Details | BINDING: BINDING => ECO:0000269|PubMed:16281028, ECO:0000269|PubMed:24462099, ECO:0000269|PubMed:27618671, ECO:0007744|PDB:2A5S, ECO:0007744|PDB:2A5T, ECO:0007744|PDB:4NF4, ECO:0007744|PDB:4NF8, ECO:0007744|PDB:5I56, ECO:0007744|PDB:5I57, ECO:0007744|PDB:5I58, ECO:0007744|PDB:5I59, ECO:0007744|PDB:5JTY |
Chain | Residue | Details |
B | ARG121 | |
A | ILE159 | |
A | TYR203 |
site_id | SWS_FT_FI3 |
Number of Residues | 2 |
Details | BINDING: BINDING => ECO:0000269|PubMed:16281028, ECO:0000269|PubMed:24462099, ECO:0007744|PDB:2A5S, ECO:0007744|PDB:2A5T, ECO:0007744|PDB:4NF4, ECO:0007744|PDB:4NF8 |
Chain | Residue | Details |
B | SER173 | |
B | TYR214 |
site_id | SWS_FT_FI4 |
Number of Residues | 3 |
Details | CARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255 |
Chain | Residue | Details |
B | ASN46 | |
B | ASN47 | |
B | ASN171 |
site_id | SWS_FT_FI5 |
Number of Residues | 1 |
Details | CARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0007744|PubMed:24090084 |
Chain | Residue | Details |
A | GLY242 |