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5JI0

PPARgamma-RXRalpha(S427F) heterodimer in complex with SRC-1, rosiglitazone, and 9-cis-retanoic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003707molecular_functionnuclear steroid receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0005634cellular_componentnucleus
D0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue 9CR A 501
ChainResidue
AILE268
AGLN275
ATRP305
APHE313
AARG316
ALEU326
AALA327
ACYS432
ALEU436

site_idAC2
Number of Residues12
Detailsbinding site for residue BRL D 501
ChainResidue
DPHE282
DCYS285
DGLN286
DSER289
DHIS323
DTYR327
DILE341
DMET364
DHIS449
DLEU453
DTYR473
DHOH768

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ESER698
FSER698
DHIS449
DTYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
DLYS224

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: Phosphoserine; by MAPK8 and MAPK9 => ECO:0000250|UniProtKB:P28700
ChainResidueDetails
ASER260

224201

PDB entries from 2024-08-28

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