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5J0D

Crystal structure of the bromodomain of human CREBBP in complex with a benzoxazepine compound

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 6F9 A 1201
ChainResidue
ALEU1109
AGLN1187
AEDO1204
AHOH1302
AHOH1306
AHOH1307
AHOH1375
APRO1110
APHE1111
AVAL1115
ALEU1120
AASN1168
AARG1173
AVAL1174
APHE1177

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 1202
ChainResidue
ALYS1141
AGLN1146
AHOH1308
AHOH1342

site_idAC3
Number of Residues5
Detailsbinding site for residue EDO A 1203
ChainResidue
AGLU1107
ATRP1158
AASN1162
APHE1177
ALYS1180

site_idAC4
Number of Residues10
Detailsbinding site for residue EDO A 1204
ChainResidue
AASP1105
APRO1106
ALEU1109
ATYR1175
ASER1179
A6F91201
AHOH1302
AHOH1305
AHOH1348
AHOH1382

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

221716

PDB entries from 2024-06-26

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