Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5IG6

Ultra-high resolution crystal structure of second bromodomain of BRD2 in complex with inhibitor 6B3

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue CL A 501
ChainResidue
AGLN412
AGLN412
AARG419
AARG419

site_idAC2
Number of Residues7
Detailsbinding site for residue CL A 502
ChainResidue
AHOH678
AHOH707
ATYR386
APRO393
AMET394
AASN424
AHOH621

site_idAC3
Number of Residues5
Detailsbinding site for residue GOL A 503
ChainResidue
ATYR426
AARG440
AGLN443
AASP444
AGLU447

site_idAC4
Number of Residues9
Detailsbinding site for residue GOL A 504
ChainResidue
ATYR368
ALYS402
AASP407
AMET438
ALYS441
AHOH619
AHOH636
AHOH646
AHOH788

site_idAC5
Number of Residues11
Detailsbinding site for residue 6B3 A 505
ChainResidue
APRO371
AVAL376
ALEU381
ALEU383
AASN429
AHIS433
AHOH610
AHOH620
AHOH635
AHOH690
AHOH721

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon