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5ICJ

Crystal structure of the Mycobacterium tuberculosis transcriptional repressor EthR2 in complex with BDM41420

Functional Information from GO Data
ChainGOidnamespacecontents
A0000976molecular_functiontranscription cis-regulatory region binding
A0003677molecular_functionDNA binding
A0003700molecular_functionDNA-binding transcription factor activity
A0005886cellular_componentplasma membrane
A0006355biological_processregulation of DNA-templated transcription
B0000976molecular_functiontranscription cis-regulatory region binding
B0003677molecular_functionDNA binding
B0003700molecular_functionDNA-binding transcription factor activity
B0005886cellular_componentplasma membrane
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 69Y A 301
ChainResidue
AGLU70
ATHR138
ALEU167
AASP168
AMET77
AILE93
AALA96
ATRP100
AILE113
APHE126
AALA130
ASER134

site_idAC2
Number of Residues15
Detailsbinding site for residue 69Y B 301
ChainResidue
BGLU70
BMET74
BILE93
BALA96
BVAL97
BTRP100
BILE113
BLEU114
BPHE126
BALA130
BSER134
BTHR138
BLEU141
BLEU167
BASP168

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PDB entries from 2024-07-24

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