Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5I89

Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02857790

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue ACT A 1201
ChainResidue
APRO1114
APRO1132
AARG1140
AHOH1324
AHOH1378
AHOH1381

site_idAC2
Number of Residues6
Detailsbinding site for residue CA A 1202
ChainResidue
AHOH1422
AHOH1463
AHOH1481
AASP1105
AHOH1314
AHOH1363

site_idAC3
Number of Residues11
Detailsbinding site for residue 69B A 1203
ChainResidue
ALEU1109
APRO1110
AVAL1115
ALEU1120
ATYR1125
AASN1168
AARG1173
AVAL1174
AHOH1309
AHOH1374
AHOH1467

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

225946

PDB entries from 2024-10-09

PDB statisticsPDBj update infoContact PDBjnumon