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5I83

Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02773986

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SCN A 1201
ChainResidue
ATRP1151
ATHR1171
AMET1193
AHOH1346
AHOH1473

site_idAC2
Number of Residues10
Detailsbinding site for residue 68Y A 1202
ChainResidue
ATYR1167
AASN1168
AARG1173
AVAL1174
AHOH1312
AHOH1330
APRO1110
AVAL1115
ALEU1120
ATYR1125

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

222415

PDB entries from 2024-07-10

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