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5I1Q

Second bromodomain of TAF1 bound to a pyrrolopyridone compound

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 67C A 1701
ChainResidue
APRO1527
ATYR1582
AASN1583
ATYR1589
ATYR1601
AHOH1875
APHE1528
APRO1531
AVAL1532
AASN1533
APHE1536
AVAL1537
ATYR1540
AMET1548

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFhhpvNkkfvp..DYYkvIvnpMdletIrkniskhk..Yqsresflddvnl.IlaNSvkY
ChainResidueDetails
ASER1525-TYR1582

224931

PDB entries from 2024-09-11

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