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5HRN

HIV Integrase Catalytic Domain containing F185K mutation complexed with GSK0002

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue CAC A 301
ChainResidue
ACYS65
AGLU92
ATHR97
AASN120

site_idAC2
Number of Residues4
Detailsbinding site for residue CAC A 302
ChainResidue
ACYS130
AILE135
ALYS136
AGLN137

site_idAC3
Number of Residues6
Detailsbinding site for residue SO4 A 303
ChainResidue
AGLU170
AHIS171
ALEU172
AHOH412
AHOH481
ALYS71

site_idAC4
Number of Residues9
Detailsbinding site for residue EDO A 304
ChainResidue
AALA105
AGLY106
ATRP108
APRO109
AASN184
ALYS185
AGLY197
AHOH449
AHOH482

site_idAC5
Number of Residues3
Detailsbinding site for residue EDO A 305
ChainResidue
AGLU69
AGLY163
AHOH442

site_idAC6
Number of Residues12
Detailsbinding site for residue 65P A 306
ChainResidue
ALEU102
ATHR125
AALA129
ATRP132
AGLN168
AALA169
AGLU170
AHIS171
ATHR174
AHOH427
AHOH483
AHOH498

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000305
ChainResidueDetails
AGLU152

Catalytic Information from CSA
site_idMCSA1
Number of Residues
DetailsM-CSA 175
ChainResidueDetails

218500

PDB entries from 2024-04-17

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